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Structure Catalog Product Name CAS Molecular Formula Molecular Weight Target Inquiry
3-nitrophenothiazine BPL-100084 3-nitrophenothiazine 1628-77-9 C12H8N2O2S 244.27

Alpha-syn

 Inquiry
Deltazinone BPL-100085 Deltazinone 894554-89-3 C27H31N5O2 457.57

PDEdelta

 Inquiry
Description: Deltazinone is a highly potent and selective PDEδ inhibitor.
1-[4-[2-methyl-6-[[5-[(E)-2-(3-methylphenyl)ethenyl]-1,3-thiazol-2-yl]amino]pyrimidin-4-yl]piperazin-1-yl]hex-5-yn-1-one BPL-100086 1-[4-[2-methyl-6-[[5-[(E)-2-(3-methylphenyl)ethenyl]-1,3-thiazol-2-yl]amino]pyrimidin-4-yl]piperazin-1-yl]hex-5-yn-1-one 2512848-38-1 C27H30N6OS 486.63

BCR-ABL T315I

 Inquiry
4-[[(1S,5R)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-2-chlorobenzonitrile BPL-100087 4-[[(1S,5R)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-2-chlorobenzonitrile C14H15ClN2O 262.73

AR

 Inquiry
VPC-14228 BPL-100088 VPC-14228 19983-28-9 C13H14N2OS 246.33

AR
AR-V7

 Inquiry
Description: VPC-14228 is a specific inhibitor of AR-DBD. It acts by inhibiting both Y594A and Q592A mutants, blocking the interaction of the AR with androgen response elements in the nucleus.
N-[3-[2-[4-(4-ethylpiperazin-1-yl)anilino]thieno[3,2-d]pyrimidin-7-yl]phenyl]methanesulfonamide BPL-100089 N-[3-[2-[4-(4-ethylpiperazin-1-yl)anilino]thieno[3,2-d]pyrimidin-7-yl]phenyl]methanesulfonamide 1644557-92-5 C25H28N6O2S2 508.66

AAK1
AURKA
BMP2K
CAMKK1
CDK1
CDK16
CDK17
CDK2
CDK4
CDK6
CDK7
EIF2AK2
EIF2AK4
FER
GAK
LATS1
LCK
LIMK2
MAP3K11
MAPK6
MAPK8
MAPK9
MAPKAPK5
MARK2
MARK4
MKNK2
NEK9
PLK4
PTK2B
RPS6KB1
SIK2
SNRK
STK17A
STK17B
STK35
ULK1
ULK3
Wee1

 Inquiry
9-cyclopentyl-2-N-[4-(4-methylpiperazin-1-yl)phenyl]-8-N-phenylpurine-2,8-diamine BPL-100090 9-cyclopentyl-2-N-[4-(4-methylpiperazin-1-yl)phenyl]-8-N-phenylpurine-2,8-diamine 1350544-90-9 C27H32N8 468.61

EGFR
EGFR e19d
EGFR L858R/T790M

 Inquiry
2-[4-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl]amino]phenyl]acetonitrile BPL-100091 2-[4-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl]amino]phenyl]acetonitrile 1636166-79-4 C19H20N8 360.43

AAK1
AURKA
BMP2K
GSK3A
GSK-3beta

 Inquiry
1-[3-(3-amino-1H-indazol-4-yl)phenyl]-3-(3-propan-2-ylphenyl)urea BPL-100092 1-[3-(3-amino-1H-indazol-4-yl)phenyl]-3-(3-propan-2-ylphenyl)urea 1800110-27-3 C23H23N5O 385.47

VEGFR-2

 Inquiry
2-[4-[[4-[(4,5-dimethyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]acetonitrile BPL-100093 2-[4-[[4-[(4,5-dimethyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]acetonitrile C17H17N7 319.37

GSK3A
GSK-3beta

 Inquiry
2-[4-[[4-[(4-ethyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]acetonitrile BPL-100093 2-[4-[[4-[(4-ethyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]acetonitrile C17H17N7 319.37

GSK-3beta

 Inquiry
[8-(4-Methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-(3-piperazin-1-yl-phenyl)-amine BPL-100094 [8-(4-Methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-(3-piperazin-1-yl-phenyl)-amine 1257706-63-0 C23H24N6O2S 448.55

JAK2

 Inquiry
methyl 4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoate BPL-100094 methyl 4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoate 2541626-63-3 C22H25N5O3 407.47

CDK2
CDK4
CDK6
AAK1
AURKA
JAK2

 Inquiry
4-{[4-{[3-(methylsulfonyl)benzyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzamide BPL-100095 4-{[4-{[3-(methylsulfonyl)benzyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzamide 1073154-92-3 C20H18F3N5O3S 465.45

FAK

 Inquiry
8-(3,5-difluoropyridin-2-yl)-N,15-dimethyl-4-(methylsulfonylmethyl)-14-oxo-8,12,15-triazatetracyclo[8.6.1.0^2,7.0^13,17]heptadeca-1(16),2(7),3,5,10,13(17)-hexaene-5-carboxamide BPL-100096 8-(3,5-difluoropyridin-2-yl)-N,15-dimethyl-4-(methylsulfonylmethyl)-14-oxo-8,12,15-triazatetracyclo[8.6.1.0^2,7.0^13,17]heptadeca-1(16),2(7),3,5,10,13(17)-hexaene-5-carboxamide C24H21F2N5O4S 513.52

BRD4

 Inquiry
4-[[(3aR,6aS)-5-amino-3a,6a-dimethyl-1,2,3,4,5,6-hexahydropentalen-2-yl]oxy]-2-chlorobenzonitrile BPL-100097 4-[[(3aR,6aS)-5-amino-3a,6a-dimethyl-1,2,3,4,5,6-hexahydropentalen-2-yl]oxy]-2-chlorobenzonitrile C17H21ClN2O 304.82

AR

 Inquiry
[4-({4-[(5-Cyclopropyl-1h-Pyrazol-3-Yl)amino]pyrimidin-2-Yl}amino)phenyl]acetonitrile BPL-100098 [4-({4-[(5-Cyclopropyl-1h-Pyrazol-3-Yl)amino]pyrimidin-2-Yl}amino)phenyl]acetonitrile 1092559-18-6 C18H17N7 331.38

AAK1
AURKA
AURKB
BMP2K
CDK9
EPHB2
GSK-3beta
ITK
LATS1
MAP4K2
NEK9
PAK4
PLK4
STK17B

 Inquiry
3-[3-[4-(aminomethyl)phenyl]-5-phenylimidazo[4,5-b]pyridin-2-yl]pyridin-2-amine BPL-100099 3-[3-[4-(aminomethyl)phenyl]-5-phenylimidazo[4,5-b]pyridin-2-yl]pyridin-2-amine 1313881-75-2 C24H20N6 392.47

AKT1
AKT2
AKT3

 Inquiry
methyl 4-[5-ethoxy-1-methyl-6-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]benzimidazol-2-yl]-2,2-dimethylbutanoate BPL-100100 methyl 4-[5-ethoxy-1-methyl-6-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]benzimidazol-2-yl]-2,2-dimethylbutanoate 2713973-42-1 C24H27F3N4O4 492.50

IRAK4

 Inquiry
N8 Pyrido[2,3-d]pyrimidin-7-one deriv. 48 BPL-100101 N8 Pyrido[2,3-d]pyrimidin-7-one deriv. 48 211247-20-0 C20H20N4O 332.41

AAK1
AURKA
AURKB
CDK6
CDK9
FGFR2
STK17A
TTK

 Inquiry

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